Basic Information
ID: ALA4351620
Type: Binding
Description: Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by HTRF assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Histone acetyltransferase PCAF(ALA5500)
Document: ALA4350961
Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by HTRF assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4351620
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 421.42 | 3.06 | 3.06 |
| 443.55 | 3.74 | 3.74 |
| 413.53 | 3.83 | 3.83 |
| 367.45 | 2.17 | 2.17 |
| 393.54 | 3.50 | 3.50 |
| 387.49 | 3.31 | 3.31 |
| 337.43 | 2.16 | 2.16 |
| 439.87 | 3.83 | 3.83 |
| 287.37 | 1.35 | 1.35 |
| 429.52 | 3.95 | 3.95 |
| 416.32 | 2.92 | 2.92 |
| 301.39 | 1.69 | 1.69 |
| 353.43 | 1.87 | 1.87 |
| 360.47 | 3.69 | 3.69 |
| 395.46 | 1.93 | 1.93 |