Basic Information
ID: ALA4352690
Type: Binding
Description: Positive allosteric modulation of human CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced beta-arrestin recruitment preincubated for 30 mins followed by CP55940 addition and measured after 90 to 180 mins by PathHunter assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA4350967
Positive allosteric modulation of human CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced beta-arrestin recruitment preincubated for 30 mins followed by CP55940 addition and measured after 90 to 180 mins by PathHunter assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4352690
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 431.45 | 7.99 | 7.99 |
| 429.46 | 6.77 | 6.77 |
| 362.45 | 5.61 | 5.61 |
| 413.46 | 7.18 | 7.18 |
| 416.42 | 6.32 | 6.32 |
| 356.86 | 6.53 | 6.53 |
| 373.44 | 5.18 | 5.18 |
| 382.87 | 5.96 | 5.96 |
| 439.42 | 8.00 | 8.00 |
| 396.44 | 6.85 | 6.85 |
| 396.44 | 6.85 | 6.85 |
| 396.44 | 6.85 | 6.85 |