ID: ALA4352702
Type: Functional
Description: Positive allosteric modulation of human Gi/Go-coupled CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimulated cAMP production preincubated for 30 mins followed by CP55940 addition and measured after 30 to 60 mins by Hit-hunter assay relative to CP55940
Format: BAO_0000219
Organism: Homo sapiens
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA4350967
Positive allosteric modulation of human Gi/Go-coupled CB1 receptor expressed in CHOK1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimulated cAMP production preincubated for 30 mins followed by CP55940 addition and measured after 30 to 60 mins by Hit-hunter assay relative to CP55940: 1
Bioactivity
Activity Types for Assay ALA4352702
Emax
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
362.45 | 5.61 | 5.61 |
373.44 | 5.18 | 5.18 |
396.44 | 6.85 | 6.85 |
396.44 | 6.85 | 6.85 |