Basic Information
ID: ALA4356375
Type: Functional
Description: Agonist activity at human H3R expressed on HEK293T cells assessed as inhibition of forskolin-induced CRE-driven luciferase activity co-incubated with forskolin for 6 hrs and measured after 30 mins by CRE-luciferase reporter gene assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4356375
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 111.15 | -0.09 | -0.09 |
| 235.34 | 0.98 | 0.98 |
| 341.37 | 0.25 | 0.25 |
| 207.28 | 0.33 | 0.33 |
| 309.33 | -0.19 | -0.19 |
| 281.27 | -0.79 | -0.79 |
| 193.25 | -0.23 | -0.23 |
| 221.31 | 0.37 | 0.37 |
| 295.30 | -0.53 | -0.53 |
| 266.18 | -0.22 | -0.22 |
| 179.23 | -0.49 | -0.49 |
| 207.28 | 0.17 | 0.17 |
| 221.31 | 0.59 | 0.59 |
| 323.35 | 0.25 | 0.25 |
| 337.38 | 0.64 | 0.64 |
| 235.34 | 0.93 | 0.93 |
| 309.33 | -0.14 | -0.14 |
| 207.28 | 0.03 | 0.03 |
| 335.36 | 0.34 | 0.34 |
| 337.38 | 0.59 | 0.59 |
| 337.38 | 0.64 | 0.64 |
| 221.31 | 0.42 | 0.42 |
| 207.28 | 0.12 | 0.12 |
| 337.38 | 0.49 | 0.49 |