Assay Report Card

Basic Information

ID: ALA4356489

Type: Binding

Description: Inhibition of verampil-stimulated ATPase hydrolysis in recombinant human MDR1 expressed in Pichia pastoris measured after 30 mins in presence of NADH by coupled enzyme assay (Rvb = 100 +/- 6 %)

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
519.636.016.01
516.645.595.59
626.587.617.61
534.696.936.93
458.595.195.19
557.727.597.59
541.706.386.38
542.756.226.22
574.757.047.04
586.767.607.60
574.705.805.80