Assay Report Card

Basic Information

ID: ALA4357466

Type: Functional

Description: Inverse agonist activity at human melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of basal cAMP accumulation incubated for 2 hrs by cAMP Alpha-screen assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
949.13-1.14-1.14
993.14-1.52-1.52
924.09-0.56-0.56
930.08-0.44-0.44
1005.19
896.08-0.47-0.47
977.18-0.50-0.50
965.13-1.43-1.43
958.09-0.52-0.52