Assay Report Card

Basic Information

ID: ALA4359317

Type: Binding

Description: Inhibition of N-terminal His-tagged human PPARgamma LBD (207 to 474 residues) expressed in Escherichia coli Rosetta (DE3) pLysS assessed as S245 phosphorylation level at 10 uM by phospho gel stain method relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
357.442.492.49
527.505.995.99
318.374.434.43
308.382.272.27
321.423.633.63