Basic Information
ID: ALA4359586
Type: Binding
Description: Displacement of Alexa Fluor 647-labeled ligand from BRD4 BD1 Y390A mutant (1 to 477 residue) (unknown origin) measured after 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4359586
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 494.37 | 3.03 | 3.03 |
| 497.42 | 1.70 | 1.70 |
| 428.31 | 1.71 | 1.71 |
| 397.80 | 0.26 | 0.26 |
| 457.94 | 0.40 | 0.40 |
| 478.37 | 2.86 | 2.86 |
| 513.41 | 2.14 | 2.14 |
| 399.86 | 1.21 | 1.21 |
| 428.90 | 1.39 | 1.39 |
| 414.87 | 1.00 | 1.00 |
| 414.87 | 1.00 | 1.00 |
| 472.37 | 1.86 | 1.86 |
| 385.87 | 1.69 | 1.69 |
| 414.87 | 0.86 | 0.86 |
| 525.43 | 1.61 | 1.61 |
| 497.42 | 1.70 | 1.70 |
| 428.90 | 1.25 | 1.25 |
| 426.88 | 1.00 | 1.00 |
| 444.90 | 0.49 | 0.49 |
| 428.90 | 1.11 | 1.11 |
| 523.46 | 2.09 | 2.09 |
| 470.39 | 2.66 | 2.66 |
| 478.37 | 3.80 | 3.80 |
| 414.87 | 1.00 | 1.00 |
| 525.47 | 2.48 | 2.48 |
| 511.45 | 2.09 | 2.09 |
| 440.91 | 1.25 | 1.25 |
| 477.38 | 4.41 | 4.41 |
| 374.81 | 0.08 | 0.08 |
| 470.39 | 2.66 | 2.66 |
| 565.42 | 2.63 | 2.63 |
| 485.41 | 1.77 | 1.77 |
| 479.01 | 1.98 | 1.98 |
| 485.41 | 1.77 | 1.77 |
| 413.88 | 1.94 | 1.94 |
| 428.90 | 1.39 | 1.39 |
| 414.87 | 0.86 | 0.86 |
| 523.46 | 2.09 | 2.09 |
| 483.39 | 1.36 | 1.36 |
| 428.90 | 1.11 | 1.11 |
| 499.39 | 1.89 | 1.89 |
| 302.78 | 2.08 | 2.08 |
| 428.90 | 1.25 | 1.25 |
| 527.44 | 2.38 | 2.38 |
| 479.01 | 1.98 | 1.98 |
| 401.83 | 1.04 | 1.04 |
| 454.94 | 1.78 | 1.78 |
| 472.37 | 1.86 | 1.86 |
| 493.38 | 2.76 | 2.76 |
| 513.41 | 2.14 | 2.14 |
| 456.37 | 2.33 | 2.33 |