Assay Report Card

Basic Information

ID: ALA4359941

Type: ADME

Description: Inhibition of human recombinant full length N-terminal His6-tagged IRAK1 (Argl94 to Ser712 residues) expressed in insect cells using H-KKARFSRFAGSSPSQSSMVAR as substrate incubated for 60 mins by fluorescence polarisation assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
401.472.702.70
319.322.542.54
307.312.472.47
318.343.143.14
504.602.402.40
402.462.742.74
476.541.901.90
457.543.363.36
451.562.872.87
493.592.642.64
490.571.911.91
477.532.172.17
458.532.752.75
415.503.593.59
391.442.072.07
319.322.542.54
465.542.262.26
372.433.523.52