Antagonist activity at MOR in Wistar rat brain membranes at 10 uM in presence of Tyr-D-Ala-Gly-Phe-NH2 after 60 mins by [35S]-GTPgammaS binding assay ...

Basic Information

ID: ALA4360752

Type: Functional

Description: Antagonist activity at MOR in Wistar rat brain membranes at 10 uM in presence of Tyr-D-Ala-Gly-Phe-NH2 after 60 mins by [35S]-GTPgammaS binding assay relative to control

Format: BAO_0000249

Organism: Rattus norvegicus

Strain: Wistar

Tissue: Brain

Subcellular Fraction: Membranes

Target:  Mu opioid receptor(ALA270)

Document:  ALA4359826

Antagonist activity at MOR in Wistar rat brain membranes at 10 uM in presence of Tyr-D-Ala-Gly-Phe-NH2 after 60 mins by [35S]-GTPgammaS binding assay relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
327.381.301.30
958.176.516.51
797.955.685.68