Basic Information
ID: ALA4360754
Type: Binding
Description: Antagonist activity at MOR/CB1R/CB2R in Wistar rat brain membranes at 10 uM in presence of N-[6-[[2-[[(4R,4aS,7aR,12bS)-4a-hydroxy-9-methoxy-3-methyl-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-ylidene]amino]oxyacetyl]amino]hexyl]-6-[3-(naphthalene-1-carbonyl)indol-1-yl]hexanamide after 60 mins by [35S]-GTPgammaS binding assay relative to control
Organism: Rattus norvegicus
Strain: Wistar
Tissue: Brain
Subcellular Fraction: Membranes
Activity Charts
Bioactivity
Activity Types for Assay ALA4360754
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 958.17 | 6.51 | 6.51 |
| 797.95 | 5.68 | 5.68 |