Basic Information
ID: ALA4360755
Type: Binding
Description: Antagonist activity at MOR/CB1R/CB2R in Wistar rat brain membranes at 10 uM in presence of (S)-N-((2R,8S)-18-(3-(1-naphthoyl)-1H-indol-1-yl)-8-benzyl-3,6,9,12-tetraoxo-4,7,10,13-tetraazaoctadecan-2-yl)-2-amino-3-(4-hydroxyphenyl)propanamide after 60 mins by liquid scintillation analysis relative to control
Organism: Rattus norvegicus
Strain: Wistar
Tissue: Brain
Subcellular Fraction: Membranes
Activity Charts
Bioactivity
Activity Types for Assay ALA4360755
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 958.17 | 6.51 | 6.51 |
| 797.95 | 5.68 | 5.68 |