Assay Report Card

Basic Information

ID: ALA4361398

Type: Binding

Description: Inhibition of PCSK9 (unknown origin) interaction with LDLR expressed in human HepG2 cells assessed as LDL uptake level at 0.1 uM measured after 2 hrs by LDL-Dylight 550 dye based fluorescence assay (Rvb = 34.8 to 67%)

Organism: Homo sapiens

Cell type: HepG2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
509.665.265.26