Basic Information
ID: ALA4361688
Type: Binding
Description: Agonist activity at human alpha4beta2 nAChR expressed in GH4C1 cells assessed as increase in inward channel current measured after 3 to 4 days at -70 mV holding potential by patch clamp assay relative to acetylcholine
Format: BAO_0000219
Organism: Homo sapiens
Target: Neuronal acetylcholine receptor; alpha4/beta2(ALA1907589)
Document: ALA4359847
Agonist activity at human alpha4beta2 nAChR expressed in GH4C1 cells assessed as increase in inward channel current measured after 3 to 4 days at -70 mV holding potential by patch clamp assay relative to acetylcholine: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4361688
Imax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 328.80 | 2.54 | 2.54 |
| 312.35 | 2.02 | 2.02 |
| 324.38 | 1.89 | 1.89 |