Basic Information
ID: ALA4361764
Type: Binding
Description: Inhibition of p300 in human U2932 cells assessed as reduction in H3K27 acetylation at 10 uM measured after 4 days in presence of EZH2 inhibitor EPZ6438 by Western blot analysis
Organism: Homo sapiens
Cell type: U2932
Activity Charts
Bioactivity
Activity Types for Assay ALA4361764
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 445.43 | 4.98 | 4.98 |
| 468.43 | 6.09 | 6.09 |
| 476.40 | 6.37 | 6.37 |
| 456.38 | 5.35 | 5.35 |
| 461.50 | 5.44 | 5.44 |
| 430.36 | 5.67 | 5.67 |
| 510.54 | 6.95 | 6.95 |
| 426.43 | 4.58 | 4.58 |
| 434.40 | 4.87 | 4.87 |
| 453.40 | 5.26 | 5.26 |