Basic Information
ID: ALA4367884
Type: Binding
Description: Antagonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arrestin recruitment pretreated with non-selective cannabinoid receptor agonist CP55940 for 30 mins and measured after 20 mins by Tango assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA4364306
Antagonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arrestin recruitment pretreated with non-selective cannabinoid receptor agonist CP55940 for 30 mins and measured after 20 mins by Tango assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4367884
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 268.34 | 3.23 | 3.23 |
| 302.79 | 3.88 | 3.88 |
| 382.57 | 5.54 | 5.54 |
| 274.39 | 3.61 | 3.61 |
| 308.41 | 4.05 | 4.05 |
| 314.45 | 4.43 | 4.43 |
| 348.47 | 4.93 | 4.93 |
| 286.40 | 3.79 | 3.79 |
| 352.50 | 4.82 | 4.82 |
| 308.41 | 4.10 | 4.10 |
| 288.37 | 2.59 | 2.59 |
| 286.40 | 3.57 | 3.57 |
| 246.34 | 2.69 | 2.69 |
| 326.40 | 4.19 | 4.19 |
| 342.85 | 4.70 | 4.70 |
| 304.37 | 4.70 | 4.70 |
| 302.44 | 4.43 | 4.43 |
| 290.43 | 3.46 | 3.46 |
| 274.39 | 3.65 | 3.65 |
| 312.44 | 4.45 | 4.45 |
| 258.35 | 3.01 | 3.01 |
| 322.31 | 4.57 | 4.57 |
| 300.43 | 4.18 | 4.18 |
| 322.31 | 4.57 | 4.57 |
| 304.37 | 4.70 | 4.70 |
| 312.44 | 3.99 | 3.99 |
| 304.37 | 4.70 | 4.70 |
| 374.51 | 5.79 | 5.79 |
| 392.45 | 5.65 | 5.65 |
| 332.51 | 4.45 | 4.45 |
| 326.40 | 4.19 | 4.19 |
| 392.45 | 5.65 | 5.65 |