Basic Information
ID: ALA4369923
Type: Binding
Description: Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from human A2A adenosine receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by scintillation proximity assay relative to adenosine 5-N-ethyluronamide
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4369923
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 244.21 | -3.01 | -3.01 |
| 281.23 | -1.89 | -1.89 |
| 431.97 | 3.55 | 3.55 |
| 399.50 | 1.48 | 1.48 |
| 433.58 | 2.58 | 2.58 |
| 433.94 | 2.14 | 2.14 |
| 269.26 | -1.66 | -1.66 |
| 403.91 | 2.77 | 2.77 |
| 254.25 | -2.35 | -2.35 |
| 404.90 | 1.96 | 1.96 |
| 452.39 | 3.38 | 3.38 |
| 487.99 | 3.72 | 3.72 |
| 417.94 | 2.73 | 2.73 |
| 424.33 | 2.60 | 2.60 |
| 475.98 | 2.71 | 2.71 |
| 544.10 | 5.07 | 5.07 |