Basic Information
ID: ALA4370422
Type: Binding
Description: Displacement of BODIPY-labeled-5-((2Z)-2-((1-(difluoroboryl)-3,5-dimethyl-1H-pyrrol-2-yl)-methylene)-2H-pyrrol-5-yl)-N-(2-((3,5-difluoro-4-(trimethylsilyl)-phenyl)amino)-1-(4-(methoxymethyl)phenyl)-2-oxoethyl)-pentanamide from human His-tagged RORgammaT after 120 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4370422
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 483.54 | 3.77 | 3.77 |
| 572.66 | 4.37 | 4.37 |
| 426.49 | 2.85 | 2.85 |
| 500.60 | 4.14 | 4.14 |
| 465.94 | 4.41 | 4.41 |
| 540.54 | 4.64 | 4.64 |
| 431.49 | 3.75 | 3.75 |
| 486.57 | 3.75 | 3.75 |
| 461.52 | 3.76 | 3.76 |
| 461.52 | 3.76 | 3.76 |