Basic Information
ID: ALA4370538
Type: Binding
Description: Inhibition of recombinant human LSD1 (172 to 852 residues) using biotin-labelled H3K4me2 (1 to 24 residues) after 1 hr by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4370538
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 133.19 | 1.50 | 1.50 |
| 415.51 | 3.80 | 3.80 |
| 364.49 | 3.74 | 3.74 |
| 446.54 | 5.66 | 5.66 |
| 468.50 | 5.19 | 5.19 |
| 432.51 | 4.91 | 4.91 |
| 446.54 | 5.66 | 5.66 |
| 446.54 | 5.66 | 5.66 |
| 460.57 | 5.91 | 5.91 |
| 432.51 | 4.91 | 4.91 |
| 446.54 | 5.66 | 5.66 |
| 482.52 | 5.94 | 5.94 |
| 460.57 | 5.91 | 5.91 |
| 496.55 | 6.19 | 6.19 |
| 446.54 | 5.16 | 5.16 |
| 446.54 | 5.16 | 5.16 |
| 482.52 | 5.94 | 5.94 |
| 482.52 | 5.44 | 5.44 |