Basic Information
ID: ALA4371698
Type: Binding
Description: Displacement of [3H]-CCR2-RA-[R] from human TEV protease site linked CCR2b expressed in human U20S cell membranes co-expressing Gal4-VP16 transcription factor at 1 uM after 120 mins by scintillation spectrometry relative to control
Format: BAO_0000219
Organism: Homo sapiens
Target: C-C chemokine receptor type 2(ALA4015)
Document: ALA4371011
Displacement of [3H]-CCR2-RA-[R] from human TEV protease site linked CCR2b expressed in human U20S cell membranes co-expressing Gal4-VP16 transcription factor at 1 uM after 120 mins by scintillation spectrometry relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4371698
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 337.38 | 3.49 | 3.49 |
| 495.14 | 5.23 | 5.23 |
| 343.42 | 3.67 | 3.67 |
| 307.35 | 3.48 | 3.48 |
| 386.25 | 4.25 | 4.25 |
| 317.36 | 3.52 | 3.52 |
| 357.45 | 4.05 | 4.05 |
| 375.47 | 4.99 | 4.99 |
| 321.38 | 3.79 | 3.79 |
| 341.79 | 4.14 | 4.14 |
| 337.38 | 3.49 | 3.49 |
| 321.38 | 3.79 | 3.79 |
| 299.37 | 3.38 | 3.38 |