Assay Report Card

Basic Information

ID: ALA4372250

Type: Binding

Description: Inhibition of thermolysin activated recombinant human C-terminal 10-His tagged KLK7 (E23 to H252 residues) using MOCAc-Arg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 as substrate preincubated for 10 mins followed by substrate addition and measured after 30 mins by fluorescence analysis

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
359.483.313.31
387.893.943.94
371.443.393.39
387.893.903.90
452.764.364.36
371.443.393.39
367.473.563.56
353.453.253.25
422.344.564.56
277.351.511.51
381.503.893.89
421.574.814.81
432.344.014.01
378.463.123.12
353.453.253.25
323.834.414.41
387.893.903.90
367.473.643.64
373.873.593.59
387.893.903.90
373.873.593.59