Assay Report Card

Basic Information

ID: ALA4373579

Type: Binding

Description: Inhibition of recombinant human N-terminal GST/His6-tagged c-KIT (T544 to V976 residues) expressed in sf9 cells assessed as equivalents of test compound required to show 50% inhibition using Poly(Glu,Tyr) 4:1 as substrate after 60 mins in presence of [gamma33P]-ATP by scintillation counting method

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
563.486.616.61
494.596.176.17