ID: ALA4374439
Type: Binding
Description: Inhibition of recombinant human C-terminal 10-His tagged hepsin (Arg45 to Leu417) expressed in mouse myeloma cells using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence based assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4374439
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
652.91 | 3.90 | 3.90 |
677.63 | 3.83 | 3.83 |
419.57 | 3.76 | 3.76 |
721.80 | 3.65 | 3.65 |
687.74 | 2.38 | 2.38 |
850.34 | 3.88 | 3.88 |
735.83 | 4.11 | 4.11 |
737.82 | 2.18 | 2.18 |
702.88 | 0.14 | 0.14 |
785.87 | 3.22 | 3.22 |
749.86 | 3.98 | 3.98 |
735.83 | 3.73 | 3.73 |
875.86 | 3.04 | 3.04 |
761.87 | 4.57 | 4.57 |
791.89 | 4.38 | 4.38 |
803.86 | 3.36 | 3.36 |
661.83 | -0.13 | -0.13 |
820.31 | 3.87 | 3.87 |
803.86 | 3.36 | 3.36 |
827.95 | 4.15 | 4.15 |