Basic Information
ID: ALA4374954
Type: Binding
Description: Inhibition of bacterial N-terminal His-tagged TEV protease site linked KPC-2 (29 to 289 amino acids) expressed in Escherichia coli Transetta (DE3) preincubated for 10 mins followed by FC5 fluorescent substrate addition by fluorescence assay
Format: BAO_0000019
Organism: Bacteria
Target: Unchecked(ALA612545)
Document: ALA4373692
Inhibition of bacterial N-terminal His-tagged TEV protease site linked KPC-2 (29 to 289 amino acids) expressed in Escherichia coli Transetta (DE3) preincubated for 10 mins followed by FC5 fluorescent substrate addition by fluorescence assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4374954
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 300.30 | -1.52 | -1.52 |
| 217.29 | 0.63 | 0.63 |
| 219.12 | ||
| 307.18 | ||
| 239.10 | ||
| 303.19 | ||
| 219.12 | ||
| 177.03 | ||
| 303.19 | ||
| 343.26 | ||
| 271.12 | ||
| 267.16 | ||
| 293.15 | ||
| 267.16 | ||
| 307.18 | ||
| 358.27 | ||
| 267.16 | ||
| 297.19 | ||
| 221.06 | ||
| 253.13 | ||
| 233.14 | ||
| 279.13 | ||
| 398.25 | ||
| 267.16 | ||
| 253.13 | ||
| 253.13 | ||
| 297.19 | ||
| 235.09 | ||
| 285.15 | ||
| 271.12 | ||
| 233.14 | ||
| 177.22 | -0.25 | -0.25 |
| 285.15 | ||
| 144.97 | ||
| 130.94 |