Assay Report Card

Basic Information

ID: ALA4375692

Type: ADME

Description: Ratio of compound effect for substrate activity at PEPT1 in Sprague-Dawley rat jejunum assessed as effective permeability in absence of non-metabolized PEPT1 substrate Gly-Sar to compound effect for substrate activity at PEPT1 in Sprague-Dawley rat jejunum assessed as effective permeability in presence of non-metabolized PEPT1 substrate Gly-Sar

Organism: Rattus norvegicus

Strain: Sprague-Dawley

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
200.19-2.56-2.56
218.21-2.73-2.73
299.33-2.03-2.03