Basic Information
ID: ALA4376067
Type: Binding
Description: Inhibition of Cys5-LDEETGEFL-NH2 binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) measured after 10 to 15 mins by fluorescence polarization assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4376067
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 344.85 | 5.38 | 5.38 |
| 34.01 | 0.02 | 0.02 |
| 212.25 | 3.04 | 3.04 |
| 461.50 | 4.16 | 4.16 |
| 207.19 | -1.32 | -1.32 |
| 446.50 | 3.30 | 3.30 |
| 497.52 | 3.97 | 3.97 |
| 498.58 | 4.46 | 4.46 |
| 486.44 | 4.27 | 4.27 |
| 443.24 | 4.41 | 4.41 |
| 440.55 | 4.74 | 4.74 |
| 614.65 | 3.42 | 3.42 |
| 1052.10 | ||
| 280.26 | 3.42 | 3.42 |
| 392.16 | 3.45 | 3.45 |
| 612.69 | 2.22 | 2.22 |
| 550.64 | 3.86 | 3.86 |
| 452.58 | 4.79 | 4.79 |
| 623.71 | 5.06 | 5.06 |
| 285.26 | 2.05 | 2.05 |
| 373.42 | 5.22 | 5.22 |
| 455.50 | 5.45 | 5.45 |
| 463.62 | 5.90 | 5.90 |
| 1094.14 | ||
| 358.31 | 2.11 | 2.11 |