Basic Information
ID: ALA4376072
Type: Binding
Description: Inhibition of FAM-LDEETGEFL-NH2 binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) measured after 30 to 60 mins in absence of TCEP buffer by fluorescence polarization assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4376072
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 486.44 | 4.27 | 4.27 |
| 443.24 | 4.41 | 4.41 |
| 440.55 | 4.74 | 4.74 |
| 392.16 | 3.45 | 3.45 |