Assay Report Card

Basic Information

ID: ALA4376092

Type: Binding

Description: Ratio of IC50 for inhibition of Cys5-LDEETGEFL-NH2 binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) in absence of 0.01% Triton X-100 to IC50 for inhibition of Cys5-LDEETGEFL-NH2 binding to recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3) in presence of 0.01% Triton X-100

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
498.584.464.46
612.692.222.22