Basic Information
ID: ALA4380046
Type: Binding
Description: Displacement of Alexa647-labeled MRL-87 from human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) measured after 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4380046
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 444.80 | 5.76 | 5.76 |
| 431.30 | 5.77 | 5.77 |
| 461.83 | 6.32 | 6.32 |