Assay Report Card

Basic Information

ID: ALA4380478

Type: Binding

Description: Inhibition of human N-terminal His-tagged MLL1 complex (MLL1/Ash2L/RbBP5/WDR5/DPY-30)-mediated HMT activity using oligonucleosome as substrate preincubated for 15 mins followed by [3H]-SAM addition after 1 hr

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
488.564.424.42
458.544.414.41
476.534.554.55
540.645.485.48
501.564.944.94
515.594.084.08
486.575.115.11
476.985.365.36
503.025.635.63
512.515.305.30
519.645.505.50
501.605.495.49
456.575.025.02
501.605.595.59
497.405.715.71
428.514.404.40
442.544.714.71
462.965.055.05
460.534.854.85
514.604.684.68
497.405.715.71