Assay Report Card

Basic Information

ID: ALA4381862

Type: Binding

Description: Antagonist activity at rat alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at 10 nM at -70 mV holding potential preincubated for 5 mins followed by compound washout by two electrode voltage-clamp assay

Organism: Rattus norvegicus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
3360.72
3452.96