Basic Information
ID: ALA4385972
Type: Binding
Description: Inhibition of recombinant human FLT3 (564 to end residues) using EAIYAAPFAKKK as substrate measured after 40 mins in presence of [gamma-33P]-ATP by scintillation counting analysis
Format: BAO_0000357
Organism: Homo sapiens
Target: Tyrosine-protein kinase receptor FLT3(ALA1974)
Document: ALA4385604
Inhibition of recombinant human FLT3 (564 to end residues) using EAIYAAPFAKKK as substrate measured after 40 mins in presence of [gamma-33P]-ATP by scintillation counting analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4385972
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 560.68 | 5.86 | 5.86 |
| 433.52 | 5.19 | 5.19 |
| 444.50 | 4.52 | 4.52 |
| 581.70 | 3.19 | 3.19 |
| 481.53 | 4.79 | 4.79 |
| 431.50 | 4.80 | 4.80 |
| 430.47 | 4.13 | 4.13 |
| 503.61 | 3.52 | 3.52 |
| 433.52 | 5.02 | 5.02 |
| 473.58 | 5.97 | 5.97 |
| 447.54 | 5.41 | 5.41 |
| 603.73 | 5.16 | 5.16 |
| 449.49 | 4.94 | 4.94 |
| 459.55 | 5.58 | 5.58 |
| 429.48 | 4.24 | 4.24 |
| 448.46 | 4.27 | 4.27 |
| 459.55 | 5.58 | 5.58 |
| 462.49 | 4.66 | 4.66 |
| 462.56 | 4.17 | 4.17 |
| 447.47 | 4.38 | 4.38 |
| 504.60 | 3.94 | 3.94 |
| 391.44 | 4.14 | 4.14 |
| 491.55 | 5.39 | 5.39 |
| 459.55 | 5.73 | 5.73 |
| 467.51 | 4.40 | 4.40 |
| 475.60 | 6.19 | 6.19 |
| 443.51 | 4.63 | 4.63 |
| 463.54 | 4.38 | 4.38 |
| 409.43 | 4.28 | 4.28 |
| 481.56 | 5.66 | 5.66 |
| 457.54 | 5.02 | 5.02 |
| 463.54 | 4.65 | 4.65 |
| 405.46 | 4.15 | 4.15 |
| 463.52 | 5.33 | 5.33 |
| 445.53 | 5.19 | 5.19 |
| 518.62 | 4.33 | 4.33 |
| 419.49 | 4.63 | 4.63 |
| 449.52 | 4.26 | 4.26 |
| 490.57 | 4.92 | 4.92 |
| 445.53 | 5.19 | 5.19 |