Assay Report Card

Basic Information

ID: ALA4386410

Type: ADME

Description: Inhibition of human recombinant full length C-terminal His-tagged HDAC3 (1 to 428 residues)/N-terminal GST-tagged NCOR2 (395 to 489 residues) expressed in baculovirus infected insect cells measured after 40 mins by HDAC-Glo1/2 luminescent assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
264.322.472.47
335.412.802.80
335.412.802.80
296.332.822.82
294.353.433.43
323.402.872.87
324.382.272.27
322.362.882.88
349.433.583.58
346.393.213.21
349.433.403.40