Assay Report Card

Basic Information

ID: ALA4386538

Type: Binding

Description: Inhibition of c-KIT V560-L576 deletion/V654A double mutant phosphorylation in human GIST430 cells at 10 to 100 nM measured after 24 to 72 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: GIST430

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
519.644.684.68