Assay Report Card

Basic Information

ID: ALA4386799

Type: Binding

Description: Trans-stimulation of human LAT1 expressed in TREx HEK293 cells assessed as induction of [3H]-gabapentin efflux at 200 uM after 3 mins by scintillation counting analysis relative to L-phenylalanine

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
155.16-0.64-0.64
204.231.121.12
174.20-1.34-1.34
169.18-0.63-0.63
245.280.890.89
166.180.040.04
166.180.040.04
166.180.040.04
232.240.360.36
246.270.280.28
156.14-1.31-1.31
206.21-0.16-0.16
186.17-1.82-1.82
246.270.280.28
170.17-1.00-1.00
170.17-1.23-1.23