Assay Report Card

Basic Information

ID: ALA4387250

Type: Binding

Description: Inhibition of recombinant full length human His-tagged GRK2 expressed in baculovirus expression system at 0.1 uM using serine/threonine-16 peptide as substrate incubated for 60 mins by Z'-LYTE assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
506.614.944.94
462.584.054.05