Assay Report Card

Basic Information

ID: ALA4387484

Type: Binding

Description: Binding affinity to N-terminal His6-tagged human SETDB1 Tudor domain (197 to 403 residues) expressed in Escherichia coli BL21(DE3)-pRARE2 cells assessed as induction of HSQC shift at 5 mM by 1H-15 N HSQC-TROSY NMR spectroscopy

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
280.350.930.93
660.78-2.65-2.65
217.231.581.58
259.311.311.31
244.301.521.52
201.231.611.61