Assay Report Card

Basic Information

ID: ALA4387495

Type: Functional

Description: In-vivo inhibition of TRPV4 in Lewis rat assessed as reduction in TRPV4 activator-induced vascular permeability by measuring Evans blue plasma extravasation at 3 mg/kg, po followed by Evans blue injection immediately after intradermal TRPV4 activator application

Organism: Rattus norvegicus

Strain: Lewis

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
541.524.724.72