Assay Report Card

Basic Information

ID: ALA4388139

Type: Binding

Description: Inhibition of TNKS/TNKS2 in human COLO320DM cells assessed as upregulation of AXIN2 expression at 0.1 uM measured after 16 hrs by Western blot analysis relative to G007-LK

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
529.974.484.48
416.472.282.28
463.372.832.83
428.922.182.18
414.942.652.65
394.481.531.53
430.461.801.80
398.482.142.14
412.471.661.66
380.492.002.00
449.383.313.31