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Inhibition of recombinant bovine enterokinase activated N-terminal His-tagged recombinant human KLK1 (19 to 262 residues) expressed in baculovirus inf...

Basic Information

ID: ALA4388470

Type: ADME

Description: Inhibition of recombinant bovine enterokinase activated N-terminal His-tagged recombinant human KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells using 3',6'-bis(prolylphenylalanylarginylamino)3H-spiro(2-benzofuran-1,9'-xanthen)-3-one;TFA as substrate measured at 30 secs interval for 5 mins by fluorescence intensity assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: Sf9

Target:  Kallikrein 1(ALA2319)

Document:  ALA4387717

Inhibition of recombinant bovine enterokinase activated N-terminal His-tagged recombinant human KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells using 3',6'-bis(prolylphenylalanylarginylamino)3H-spiro(2-benzofuran-1,9'-xanthen)-3-one;TFA as substrate measured at 30 secs interval for 5 mins by fluorescence intensity assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
418.502.882.88
387.872.342.34
291.362.972.97
375.484.154.15
279.352.472.47
378.482.912.91
404.472.632.63
293.332.112.11
336.233.113.11
431.935.215.21
251.721.311.31
409.494.014.01
424.462.102.10
407.473.763.76
431.935.215.21
265.751.321.32
434.933.953.95
410.431.841.84
398.473.953.95
397.484.554.55
325.372.772.77
295.352.472.47
381.443.373.37
435.923.343.34
431.935.215.21
265.322.462.46
388.433.543.54