Assay Report Card

Basic Information

ID: ALA4389078

Type: Binding

Description: Reversible inhibition of recombinant full-length N-terminal 6-His-tagged human BTK expressed in baculovirus infected Sf21 insect cells using fluorescent-labeled polyGAT peptide as substrate incubated for 30 mins by TR-FRET assay

Organism: Homo sapiens

Cell type: Sf21

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
468.616.286.28
372.434.264.26
446.945.645.64
495.635.985.98
481.605.595.59
397.484.594.59
446.945.645.64
479.595.795.79
413.494.384.38
446.945.645.64
378.483.783.78
436.524.704.70
412.504.994.99
413.494.384.38
480.626.646.64
352.443.753.75
430.495.135.13
348.412.982.98
430.495.135.13
409.504.964.96
452.565.865.86
412.504.994.99
481.605.595.59
430.495.135.13
411.514.524.52
544.644.204.20
338.423.363.36
412.504.994.99
480.496.006.00
413.494.384.38
372.434.074.07
464.534.434.43
433.544.144.14