Assay Report Card

Basic Information

ID: ALA4390461

Type: Binding

Description: Inverse agonist activity at human Gal4-fused RORbeta LBD (200 to 559 residues) expressed in human Jurkat cells measured after 18 hrs by steady-glo luciferase reporter gene assay

Organism: Homo sapiens

Cell type: Jurkat

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
651.574.934.93
661.635.625.62
626.575.315.31
625.535.375.37
667.584.794.79
655.565.435.43
633.584.844.84
645.546.006.00
599.545.575.57
645.546.006.00
627.555.915.91
669.637.087.08
661.635.625.62
649.583.963.96
619.554.454.45
655.606.696.69
641.586.006.00
643.555.025.02
663.614.614.61
625.535.375.37
641.586.306.30
663.614.204.20
625.535.375.37
639.566.056.05
653.596.446.44
655.606.696.69
655.565.435.43
645.546.006.00
613.575.825.82
647.615.235.23
651.585.505.50
671.605.925.92
641.586.306.30
657.585.685.68
641.586.306.30