Assay Report Card

Basic Information

ID: ALA4390491

Type: Binding

Description: Inhibition of recombinant human full-length C-terminal FLAG-tagged HDAC1 expressed in baculovirus expression system at 10 nM using Ac-peptide-AMC as substrate preincubated for 15 mins followed by substrate addition by fluorescence assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
264.322.472.47
354.463.203.20
349.433.333.33
463.542.912.91
421.513.143.14
407.482.482.48
393.452.622.62
450.552.292.29
409.451.331.33
421.513.143.14
407.482.582.58
437.502.372.37
435.533.533.53
437.502.372.37
450.552.292.29
464.572.512.51
407.482.482.48
423.482.512.51
423.481.811.81
451.532.592.59
421.512.972.97
436.521.731.73
435.533.213.21