Assay Report Card

Basic Information

ID: ALA4390495

Type: Binding

Description: Inhibition of wild-type human N-terminal GST-tagged CDK2/cycA2 expressed in Sf21 insect cells at 100 nM using FAM-labelled substrate preincubated for 10 mins followed by substrate addition and measured after 30 mins by fluorescence assay relative to control

Organism: Homo sapiens

Cell type: Sf21

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
264.322.472.47
354.463.203.20
349.433.333.33
463.542.912.91
421.513.143.14
407.482.482.48
393.452.622.62
450.552.292.29
409.451.331.33
421.513.143.14
407.482.582.58
437.502.372.37
435.533.533.53
437.502.372.37
450.552.292.29
464.572.512.51
407.482.482.48
423.482.512.51
423.481.811.81
451.532.592.59
421.512.972.97
436.521.731.73
435.533.213.21