ID: ALA4392123
Type: Binding
Description: Agonist activity at recombinant C-terminal RLuc8-fused human D1 receptor expressed in HEK29T cells co-expressing N-terminal Venus-tagged beta-arrestin2 assessed as increase in beta-arrestin2 recruitment measured after 15 mins in presence of coelenterazine H by BRET assay relative to dopamine
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4392123
Emax
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
356.39 | 4.95 | 4.95 |
341.37 | 5.24 | 5.24 |
356.39 | 4.95 | 4.95 |
438.45 | 6.20 | 6.20 |
357.37 | 4.22 | 4.22 |
346.39 | 5.31 | 5.31 |
372.45 | 5.42 | 5.42 |
411.41 | 6.42 | 6.42 |
355.40 | 4.45 | 4.45 |
395.34 | 5.95 | 5.95 |
361.40 | 5.09 | 5.09 |
363.32 | 5.21 | 5.21 |
355.40 | 4.90 | 4.90 |
316.36 | 4.20 | 4.20 |
332.36 | 4.28 | 4.28 |
342.36 | 4.52 | 4.52 |
423.52 | 6.24 | 6.24 |
410.36 | 5.66 | 5.66 |
366.42 | 5.35 | 5.35 |
331.38 | 4.88 | 4.88 |
356.39 | 4.08 | 4.08 |