Assay Report Card

Basic Information

ID: ALA4392217

Type: Binding

Description: Inhibition of human His-tagged G9a (913 to 1193 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL assessed as enzyme residual activity at 10 uM using H3-21 peptide as substrate preincubated for 10 mins in presence of SAM followed by substrate addition by fluorescence assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1087.30