Basic Information
ID: ALA4394502
Type: Binding
Description: Inhibition of 20S proteasome beta5 subunit in human RPMI8226 cell lysate using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by substrate addition and measured at 1 min interval by fluorescence assay
Organism: Homo sapiens
Subcellular Fraction: Lysate
Activity Charts
Bioactivity
Activity Types for Assay ALA4394502
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 719.92 | 2.58 | 2.58 |
| 484.75 | ||
| 824.03 | 2.20 | 2.20 |
| 370.49 | 1.32 | 1.32 |
| 814.01 | 1.54 | 1.54 |
| 735.92 | 1.56 | 1.56 |
| 779.98 | 2.18 | 2.18 |
| 974.33 | ||
| 749.95 | 2.21 | 2.21 |