Basic Information
ID: ALA4394510
Type: Binding
Description: Inhibition of tracer 5 binding to human N-terminal nano luciferase-fused GAK expressed in HEK293 cells at 5 uM measured after 2 hrs by nanoBRET assay relative to control
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Serine/threonine-protein kinase GAK(ALA4355)
Document: ALA4393671
Inhibition of tracer 5 binding to human N-terminal nano luciferase-fused GAK expressed in HEK293 cells at 5 uM measured after 2 hrs by nanoBRET assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4394510
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 581.07 | 6.14 | 6.14 |
| 379.34 | 4.42 | 4.42 |
| 438.89 | 6.37 | 6.37 |
| 392.38 | 5.05 | 5.05 |
| 439.87 | 5.76 | 5.76 |
| 458.57 | 3.93 | 3.93 |
| 392.38 | 5.33 | 5.33 |