Assay Report Card

Basic Information

ID: ALA4396010

Type: Binding

Description: Inhibition of human topoisomerase-2alpha assessed as rate of ATP hydrolysis at 40 uM using pBR322 as substrate measured up to 30 mins in presence of 0.075 mM ATP by pyruvate kinase/lactate dehydrogenase enzyme coupled assay (Rvb = 0.884 to 1.438 microM/min)

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
461.895.565.56