Assay Report Card

Basic Information

ID: ALA4396717

Type: Binding

Description: Inverse agonist activity at full length human FLAG-tagged GAL4-DBD fused PPARgamma LBD (205 to 505 residues) expressed in COS1 cells assessed as inhibition of rosiglitazone binding measured after 18 hrs by dual luciferase reporter gene assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
281.404.384.38